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OEM Ubushinwa Bwuzuye Uruganda Igiciro Cyimiti Imiti Yumuti Rivaroxaban CAS 366789-02-8

OEM Ubushinwa Bwuzuye Uruganda Igiciro Cyimiti Imiti Yumuti Rivaroxaban CAS 366789-02-8

Ibisobanuro bigufi:

Inzira ya molekulari: C.19H18ClN3O5S

Uburemere bwa molekile: 435.88

URUBANZA no: 366789-02-8


Ibicuruzwa birambuye

Ibicuruzwa

Turabizi ko dutera imbere gusa niba dushobora kwemeza byoroshye guhuriza hamwe ibiciro hamwe nibyiza bihebuje icyarimwe kubucuruzi bwa OEM Ubushinwa Bwinshi Bwuzuye Uruganda Ibiciro bya farumasi yimiti ya Rivaroxaban CAS 366789-02-8, Ibyishimo byabakiriya nintego yacu nyamukuru.Turakwishimiye gushiraho umubano wubucuruzi natwe.Kubindi bisobanuro, menya neza ko utazategereza kuvugana natwe.
Turabizi ko dutera imbere gusa niba dushobora kwemeza byoroshye guhuriza hamwe ibiciro hamwe nibyiza bihebuje icyarimwe kuriUbushinwa Rivaroxaban n'Ikigobe 59-7939, Turatekereza rwose ko dufite ubushobozi bwuzuye bwo kuguha ibicuruzwa byuzuye.Wifuzaga gukusanya impungenge muri wewe no kubaka umubano muremure wigihe kirekire.Twese dusezeranya cyane: Csame nziza, igiciro cyiza cyo kugurisha;igiciro nyacyo cyo kugurisha, ubuziranenge bwiza.

Ikoreshwa mubarwayi bakuze bafite uburyo bwo kubaga ikibuno cyangwa gusimbuza ivi kugirango birinde imiyoboro y'amaraso (VTE).

Ikoreshwa mukurinda cyangwa kugabanya imiterere ya trombose, imitsi yimbitse (DVT) hamwe na embolisme yimpyisi (PE) nyuma yo kubagwa ikibuno cyangwa ivi.

Igipimo gisabwa ni umunwa rivaroxaban 10mg, rimwe kumunsi.Rivaroxaban 10mg irashobora gufatwa nibiryo cyangwa wenyine.Rivaroxaban ibinini 15mg cyangwa 20mg bigomba gufatwa nibiryo.

bisanzwe: usp40
Suzuma: 99-102%

Inyuma: Ifu yera
Ipaki: 25kg / ingoma

Fata 4- (4-aminophenyl) morpholin-3-imwe (SM-1), (S) -N-glycidyl phthalimide (SM-2), 5-chlorothiophene-2- Formyl chloride (SM-3) ni ibikoresho byo gutangira .Nyuma ya kondegene, cycleisation, aminolysis na acylation, rivaroxaban itaboneka iraboneka, kandi rivaroxaban yarangije gutunganywa.
Gutegura: Iki gicuruzwa nikibaho gitukura cya firime.

Ibikoresho:
Intandaro ya tablet: microcrystalline selulose, sodium ya croscarmellose, monohydrate ya lactose, hypromellose, sodium lauryl sulfate, magnesium stearate
Igipfukisho: polyethylene glycol, hypromellose, dioxyde ya titanium, okiside itukura

Rivaroxaban numuti watoranijwe cyane, umunwa uhagarika ibintu Xa.Binyuze mu guhitamo cyane no guhatanira kubuza ibintu kubuntu no guhuza ibikorwa Xa hamwe na prothrombine, ongera igice cya tromboplastine igice cyakorewe (PT) hamwe nigihe cya prothrombin (aPTT) muburyo bushingiye kumupanga, bishobora guhagarika isumo ya coagulation Inzira ya endogenous na exogenous kubuza umusaruro wa trombine na trombose.Rivaroxaban ntabwo ibuza trombine (ibintu bikora Ⅱ), nta nubwo yerekanye ko igira ingaruka kuri platine
Itandukaniro ryingenzi hagati ya rivaroxaban na fondaparinux / heparin nuko bidasaba uruhare rwa antithrombine III kandi irashobora kurwanya muburyo butaziguye Xa;mugihe heparin isaba antithrombine III gukora, kandi Nta ngaruka igira kubintu Xa murwego rwa prothrombine.

Turabizi ko dutera imbere gusa niba dushobora kwemeza byoroshye guhuriza hamwe ibiciro hamwe nibyiza bihebuje icyarimwe kubucuruzi bwa OEM Ubushinwa Bwinshi Bwuzuye Uruganda Ibiciro bya farumasi yimiti ya Rivaroxaban CAS 366789-02-8, Ibyishimo byabakiriya nintego yacu nyamukuru.Turakwishimiye gushiraho umubano wubucuruzi natwe.Kubindi bisobanuro, menya neza ko utazategereza kuvugana natwe.
OEM UbushinwaUbushinwa Rivaroxaban n'Ikigobe 59-7939, Turatekereza rwose ko dufite ubushobozi bwuzuye bwo kuguha ibicuruzwa byuzuye.Wifuzaga gukusanya impungenge muri wewe no kubaka umubano muremure wigihe kirekire.Twese dusezeranya cyane: Csame nziza, igiciro cyiza cyo kugurisha;igiciro nyacyo cyo kugurisha, ubuziranenge bwiza.


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